Topical Melatonin

Anti-agingAntioxidantPM skincare

Melatonin isn't just for sleep — applied to skin overnight, it's a potent antioxidant that protects against UV-driven oxidative damage from the previous day.

EvidenceEmerging

Strong mechanism (skin's own antioxidant system). Small RCTs support reduced UV-induced skin damage, improved hydration, and post-procedure healing. Effects: 8–16 weeks for visible changes.

Skin has melatonin receptors and produces its own melatonin — but levels drop with age. Topical melatonin applied at night functions as a powerful antioxidant in skin tissue, protecting against the lingering oxidative damage from daytime UV and pollution exposure. It's especially compelling in PM routines as a counterpart to morning vitamin C. Doesn't cause sleep effects when applied to skin (negligible systemic absorption). Small but growing trial evidence for photoaging and post-procedure healing.

Form
Topical melatonin serum — increasingly common in PM-focused skincare lines (Asystem, Naissant). Often combined with peptides or HA. 0.01–0.1% concentrations.
Dose
Apply per product instructions, PM only.
Timing
PM, after cleansing, before / instead of night moisturiser.
Schedule
Nightly.
Side effects
Generally well-tolerated. Mild irritation, rare contact dermatitis.
Interactions
Generally clean topically. Negligible systemic absorption (no sleep effects).
Contraindications
Pregnancy / breastfeeding (default caution — limited data).
Lab markers
Visual / photographic skin tracking.
Food sources
Not food.

Pairs with

Topical vitamin C + SPF (AM) — morning protection, evening repair. Topical retinoids (apply melatonin after letting retinol absorb).