Goldenseal (Hydrastis canadensis)

AntimicrobialGut

A North American root rich in berberine — used as a short-term antimicrobial for gut infections, mouth sores, and sinusitis. Overharvested in the wild.

EvidenceModerate

Moderate for acute infectious diarrhea (mostly via berberine content), topical antimicrobial use, sinusitis adjunct. Effects: days.

Hydrastis canadensis is a forest root native to eastern North America, traditionally used by Cherokee and adopted into Western herbalism for infections. Its main alkaloid berberine is the same one in the berberine entry — but goldenseal also contains hydrastine and canadine, which add their own activity. Used mostly as a short-term antimicrobial for gut infections (SIBO, traveler's diarrhea adjunct), mouth sores, sinusitis, and skin issues. The plant is severely overharvested in the wild — only buy from sustainable cultivation sources.

Form
Goldenseal root extract standardised to alkaloid content. Goldenseal tincture.
Dose
500–1,000 mg root powder 3x daily, or 250–500 mg standardised extract 2x daily.
Timing
With food.
Schedule
Short-term only (5–14 days during acute use). Not for chronic daily use — can disrupt gut flora and B-vitamin absorption.
Side effects
GI upset, mouth / throat irritation (if not encapsulated). Long-term use can reduce B-vitamin absorption.
Interactions
CYP3A4 substrates — goldenseal is a potent CYP3A4 inhibitor (similar to grapefruit but stronger). Many drug interactions. Anticoagulants — mild additive. Cyclosporine, statins, calcium channel blockers — significant interactions.
Contraindications
Pregnancy (uterine stimulant, possible kernicterus in newborn). Newborn / infant. Severe hypertension. On any narrow-therapeutic-window medication without provider input.
Lab markers
Not standard.
Food sources
Not in everyday food.

Pairs with

Echinacea (classic traditional pairing for immune / infection). Berberine (similar mechanism). Oregon grape root (related berberine-rich herb).